Boc-His(Boc)-Aib-Gln(Trt)-Gly-OH

DiPetptide

ꁇNovel Building Blocks

• Chiral Alcohol

• Chiral Amine

• Chiral Aldehyde

• Other (GNP)

ꁇAlanine Series

• Substituted Ala Derivatives

• Substituted D-Ala Derivatives

• Beta-Ala Derivatives

• N-MethylAla Derivatives

• N-EthylAla Derivatives

• Deuterated Ala Derivatives

ꁇLysine Series

• Lys Derivatives

• D-Lys Derivatives

• Beta-Lys Derivatives

• N-MethylLys Derivatives

• Alpha-MethylLys Derivatives

• N-EthylLys Derivatives

• Deuterated Lys Derivatives

ꁇIsoleucine Series

• L-Alloisoleu Derivatives

• D-ILe Derivatives

• Beta-Lys Derivatives

• N-Methyl-L-Alloisoleu Derivatives Deriva

• N-Methyl-D-ILe Derivatives

• N-Methyl-ILe Derivatives

• Deuterated ILe Derivatives

ꁇArginine Series

• Arg Derivatives

• HomoArg Derivatives

• D-Arg Derivatives

• Beta-Arg Derivatives

• N-MethylArg Derivatives

• Alpha-MethylArg Derivatives

• N-EthylArg Derivatives

• Deuterated Arg Derivatives

ꁇAspartic acid/Asparagine Series

• Asp/Asn Derivatives

• D-Asp/Asn Derivatives

• Beta-Asp/Asn Derivatives

• N-MethylAsp/Asn Derivatives

• Alpha-MethylAsp/Asn Derivatives

• N-EthylAsp/Asn Derivatives

• Deuterated Asp/Asn Derivatives

ꁇGlutamic acid/Glutamine Series

• Glu/Gln Derivatives

• HomoGlu/Gln Derivatives

• D-Glu/Gln Derivatives

• Beta-Glu/Gln Derivatives

• N-MethylGlu/Gln Derivatives

• Alpha-MethylGlu/Gln Derivatives

• N-EthylGlu/Gln Derivatives

ꁇLeucine Series

• Leu Derivatives

• HomoLeu Derivatives

• D-Leu Derivatives

• Beta-Leu Derivatives

• N-MethylLeu Derivatives

• Alpha-MethylLeu Derivatives

• N-EthylLeu Derivatives

• Deuterated Leu Derivatives

ꁇSerine Series

• Ser Derivatives

• HomoSer Derivatives

• D-Ser Derivatives

• Beta-Ser Derivatives

• N-MethylSer Derivatives

• Alpha-MethylSer Derivatives

• N-EthylSer Derivatives

• Deuterated Ser Derivatives

ꁇOrnithine Series

• Orn Derivatives

• NorOrn Derivatives

• D-Orn Derivatives

• Beta-Orn Derivatives

• N-MethylOrn Derivatives

• Alpha-MethylOrn Derivatives

• N-EthylOrn Derivatives

• Deuterated Orn Derivatives

ꁇPhenylalanine Series

• Phe Derivatives

• HomoPhe Derivatives

• D-Phe Derivatives

• Beta-Phe Derivatives

• N-MethylPhe Derivatives

• Alpha-MethylPhe Derivatives

• N-EthylPhe Derivatives

• Deuterated Phe Derivatives

ꁇThreonine Series

• Thr Derivatives

• HomoThr Derivatives

• D-Thr Derivatives

• Beta-Thr Derivatives

• N-MethylThr Derivatives

• Alpha-MethylThr Derivatives

• N-EthylThr Derivatives

• Deuterated Thr Derivatives

ꁇTryptophan Series

• Try Derivatives

• HomoTry Derivatives

• D-Try Derivatives

• Beta-Try Derivatives

• N-MethylTry Derivatives

• Alpha-MethylTry Derivatives

• N-EthylTry Derivatives

• Deuterated Try Derivatives

ꁇTyrosine Series

• Tyr Derivatives

• HomoTyr Derivatives

• D-Tyr Derivatives

• Beta-Tyr Derivatives

• N-MethylTyr Derivatives

• Alpha-MethylTyr Derivatives

• N-EthylTyr Derivatives

• Deuterated Tyr Derivatives

ꁇValine Series

• Substituted Val Derivatives

• Substituted D-Val Derivatives

• Beta-Val Derivatives

• N-MethylVal Derivatives

• N-EthylVal Derivatives

• Deuterated Val Derivatives

ꁇHistidine Series

• Substituted His Derivatives

• Substituted D-His Derivatives

• Beta-His Derivatives

• N-MethylHis Derivatives

• N-EthylHis Derivatives

• Deuterated His Derivatives

ꁇCysteine Series

• Substituted Cys Derivatives

• Substituted D-Cys Derivatives

• Beta-Cys Derivatives

• N-MethylCys Derivatives

• N-EthylCys Derivatives

• Deuterated Cys Derivatives